Figure 1: Modelled seed structures derived from the telmisartan scaffold (i) the optimal telmisartan
conformer in the non-cognate PPARα_LBP (2P54); (ii) TELMS1 shows the conserved part
of the biphenyl moiety in a blue box; (iii) TELMS2 shows in a blue box the preserved
part of the nitrogen substituted fused 5-membered ring. Structures rendered in Accelrys®
[18].
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